From:  Role of insect farming as a sustainable approach for global food security and its therapeutic applications

 Bioactive compounds having pharmacological potential and their mechanism of action.

Bioactive compoundsFormulationPharmacological potentialMechanism of actionReferences
Royal jelly (peptides, fatty acids), silkworm protein (sericin and fibroin), propolis (phenolic acid)Water and liposoluble extractsAntioxidant activityScavenges free radicals and reactive oxygen species, enhances the natural antioxidant defense system[75]
Melittin, propolis (chrysin, CAPE), cantharidin, mastoparan, royal jelly (10-hydroxy-2-decanoic acid, apalbumin)Bioactive peptidesAnticancer activityInduces apoptosis, inhibits angiogenesis and metastasis, disrupts mitochondria in cancer cells[76]
Peptides like defensins, cecropins, attacins, royalisin, propolis (flavonoids, phenolics)Polyphenolic ethanol and ethanol: water extractsAntimicrobial activityBy the disruption of cell membrane, inherent low pH, and H2O2 in bee products[61, 77, 80]
Royal jelly, MRJP-2Ethanolic extractHepatoprotective activityBoosts SOD, CAT, GSH, GST, GSH-Px, regulates Bcl-2, caspase-3, reduces inflammation and cholesterol[51, 84]
Royal jelly, silk protein, bee venom proteinBioactive peptidesNeuroprotectivity activityModulates neurotransmitters like GABA, dopamine, serotonin, aids nerve repair, reduces oxidative stress in the brain[86]

CAPE: caffeic acid phenethyl ester; CAT: catalase; GABA: gamma-aminobutyric acid; GSH: glutathione; GSH-Px: glutathione peroxidase; GST: glutathione S-transferase; MRJP: major royal jelly protein; SOD: superoxide dismutase.