From:  Alpha lipoic acid: advancing insights in diabetic neuropathy through updated systematic review and meta-analysis

 Description of included studies.

Sl. No.Author nameDose, route, duration (number of subjects)Sample size (number of subjects)InterventionParametersSafetyOutcomes and conclusions
1Ziegler et al., 2011 [29]600 mg, oral route, 4 yearsControl = 224
ALA = 230
ALA, once dailyHbA1C, NIS-LL, NIS, MNCV, NSC, VPT, TSSAdverse effects were more common with ALA, yet the placebo group had a higher incidence of deaths.ALA shows improvement in NIS and NIS-LL, but MNCV and SNAP are seen. ALA slows the progression of DSPN but doesn’t improve the condition.
2Ziegler et al., 2006 [26]600 mg, 1,200 mg, 1,800 mg, oral route, 5 weeksControl = 43
ALA 600 = 45
ALA 1,200 = 47
ALA 1,800 = 46
ALA, once dailyHbA1C, NIS, NIS-LL, NSC, TSS, global satisfactionAdverse events in the treatment group were dose-dependent, with the highest incidence observed in the 1,800 mg group.ALA shows improvement in TSS, NSC, NIS, and NIS-LL parameters when compared with the placebo group.
3Reljanovic et al., 1999 [12]600 mg, 1,200 mg, oral route, 24 monthsControl = 20
ALA 600 = 27
ALA 1,200 = 18
ALAHbA1C, MNCVTreatment-related adverse effects were noted. But the overall tolerability assessment was rated as very good or good.Improvement in MNCV is seen in the ALA 1,200 mg group.
4El-Nahas et al., 2020 [30]600 mg, two times daily (1,200 mg/day) oral route for 6 monthsControl = 100
ALA = 100
ALAHbA1C, NSS, NDS, VPT, VASNausea.ALA is effective, safe, and tolerable for the treatment of DPN.
5Ruhnau et al., 1999 [31]600 mg, three times daily, oral route (1,800 mg/day) for 3 weeksControl = 12
ALA = 12
Thioctic acid (ALA)HbA1C, TSS, NDSNo adverse effects seen.Short-term treatment with oral ALA ameliorates neuropathic symptoms.
6Vijayakumar et al., 2014 [18]600 mg, oral route, 3 monthsControl = 10
ALA = 10
ALAHbA1C, MNCVNo data available.Oral ALA improves MNCV in DN patients.
7Siddique et al., 2021 [28]600 mg, oral route, 6 monthsControl = 55
ALA = 55
ALAHbA1C, TSSNo data available.Significant improvement in TSS was seen. ALA improved symptoms of neuropathy pain and enhanced QOL.
8Millan-Guerrero et al., 2018 [37]1,200 mg, oral route, 4 weeksControl = 49
ALA = 51
ALAMNCVNo adverse effects seen.No clinically significant improvement was seen.
9Tang et al., 2007 [27]600 mg, 1,200 mg, 1,800 mg, oral route, 5 weeksControl = 43
ALA 600 = 45
ALA 1,200 = 47
ALA 1,800 = 56
ALAGlobal satisfactionNausea, vomiting, and vertigo.ALA is effective in reducing neuropathic symptoms in DSPN.

ALA: alpha lipoic acid; HbA1C: glycated hemoglobin; NIS: neuropathy impairment score; NIS-LL: NIS-low limb; MNCV: motor nerve conduction velocity; NSC: neuropathy symptoms and change; TSS: total severity score; SNAP: sensory nerve action potential; VPT: vibration perception threshold; NDS: neurological disability score; NSS: neurological symptom scale; VAS: visual analogue scale; DSPN: diabetic distal symmetric polyneuropathy; DPN: diabetic peripheral neuropathy; DN: diabetic neuropathy; QOL: quality of life.