Exploration of Targeted Anti-tumor Therapy

Radionucleotide-labeled antibody	Target	USA Food and Drug Administration (FDA) approval	Reference
⁹⁰Y-ibritumomab-tiuxetan	CD20	Yes (February 2002)	[10–20]
¹³¹I-tositumomab	CD20	Yes (June 2003)	[21–24]
⁹⁰Y-epratuzumab tetraxetan	CD22	No (Only phase I/II study)	[25]
¹⁷⁷Lu-lilotomab satetraxetan	CD37	No (Only phase I/II study)	[26–30]

Declarations

Acknowledgments

We thank Kumiko Fukushima for secretarial assistance (Kumamoto University).

Author contributions

HG: Conceptualization, Writing—original draft, Writing—review & editing, Supervision. SO: Conceptualization, Writing—review & editing, Supervision. YS: Writing—review & editing. All authors read and approved the submitted version.

Conflicts of interest

The authors declare that they have no conflicts of interest.

Ethical approval

Not applicable.

Consent to participate

Not applicable.

Consent to publication

Not applicable.

Availability of data and materials

Not applicable.

Funding

Not applicable.

Copyright

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